Amicar Oral Solution Generic Name & Formulations
Legal Class
General Description
Pharmacological Class
See Also
How Supplied
Tabs—30; Oral soln—236.5mL
Manufacturer
Generic Availability
YES
Amicar Oral Solution Indications
Indications
Amicar Oral Solution Dosage and Administration
Adult
Children
Renal Impairment
Higher plasma concentrations of aminocaproic acid may occur in patients with severe renal failure.
Amicar Oral Solution Contraindications
Contraindications
Amicar Oral Solution Boxed Warnings
Not Applicable
Amicar Oral Solution Warnings/Precautions
Warnings/Precautions
Amicar Oral Solution Pharmacokinetics
Absorption
After a single oral dose of 5g, mean ± SD peak plasma concentrations (164 ± 28mcg/mL) were reached within 1.2 ± 0.45 hours.
Distribution
After oral administration, volume of distribution was estimated to be 23.1 ± 6.6 L (mean±SD).
Elimination
Renal excretion is the primary route of elimination. Terminal elimination half-life is approximately 2 hours.
Amicar Oral Solution Interactions
Interactions
Amicar Oral Solution Adverse Reactions
Adverse Reactions
Bradycardia, hypotension, GI upset, edema, headache, malaise, CNS effects, thrombosis, others; rare: myopathy.
Amicar Oral Solution Clinical Trials
See Literature
Amicar Oral Solution Note
Not Applicable
Amicar Oral Solution Patient Counseling
See Literature