Antiretroviral Formulations
| ANTIRETROVIRAL FORMULATIONS | ||||||
|---|---|---|---|---|---|---|
| Generic & Class | Brand Name | Capsules | Tablets | Liquid | Powder | IV injection |
| Non-nucleoside Reverse Transcriptase Inhibitors (NNRTIs) | ||||||
| delavirdine | Rescriptor | • | ||||
| efavirenz | Sustiva | • | • | |||
| etravirine | Intelence | • | ||||
| nevirapine | Viramune | • | • | |||
| Viramune XR* | • | |||||
| rilpivirine | Edurant | • | ||||
| Nucleoside/Nucleotide Reverse Transcriptase Inhibitors (NRTIs) | ||||||
| abacavir | Ziagen | • | • | |||
| abacavir/lamivudine | Epzicom | • | ||||
| abacavir/lamivudine/zidovudine | Trizivir | • | ||||
| didanosine | Videx | •¹ | ||||
| Videx EC** | • | |||||
| emtricitabine | Emtriva | • | • | |||
| emtricitabine/tenofovir disoproxil fumarate | Truvada | • | ||||
| lamivudine | Epivir | • | • | |||
| lamivudine/zidovudine | Combivir | • | ||||
| stavudine | Zerit | • | •¹ | |||
| tenofovir disoproxil fumarate | Viread | • | • | |||
| zidovudine | Retrovir | • | • | • | • | |
| Protease Inhibitors (PIs) | ||||||
| atazanavir | Reyataz | • | ||||
| darunavir | Prezista | • | • | |||
| fosamprenavir | Lexiva | • | • | |||
| indinavir | Crixivan | • | ||||
| lopinavir/ritonavir | Kaletra | • | • | |||
| nelfinavir | Viracept | • | •¹ | |||
| ritonavir | Norvir | • | • | • | ||
| saquinavir | Invirase | • | • | |||
| tipranavir | Aptivus | • | • | |||
| Entry/Fusion Inhibitors | ||||||
| enfuvirtide | Fuzeon | •² | ||||
| maraviroc | Selzentry | • | ||||
| Integrase Inhibitors | ||||||
| raltegravir | Isentress | •/c | ||||
| Multiclass Fixed-Dose Combination | ||||||
| efavirenz/emtricitabine/tenofovir disoproxil fumarate | Atripla | • | ||||
| emtricitabine/rilpivirine/tenofovir disoproxil fumarate | Complera | • | ||||
| elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate | Stribild | • | ||||
| NOTES | ||||||
|
* Viramune XR = extended release tablets ** Videx EC = enteric coated delayed-release capsules. ¹ Powder for oral solution ² Powder for subcutaneous injection c = chewable tablets For a list of antiretroviral monographs, visit www.eMPR.com. (Rev. 4/2013) |
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